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Metronidazole

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CAS: 443-48-1

1.Metronidazole bụ ọgwụ nje nitroimidazole, nke a makwaara dị ka methotrexate, metronidazole, metronidazole, metronidazole, methotrexate, microorganisms anaerobic nwere mmetụta igbu egbu, ọ na-ebelata n'ime ahụ mmadụ mgbe metabolites emepụtara nwekwara mmetụta mgbochi anaerobic bacterial, na-egbochi ya. njikọ nke deoxyribonucleic acid nke nje bacteria, si otú ahụ na-egbochi uto nke nje bacteria, mmeputakwa, na n'ikpeazụ kpatara ọnwụ nje, anti-anaerobic bacteria Pu gụnyere: Bacteroides fragilis, Clostridium (n'ihi The anti-anaerobic bacteria gụnyere: Bacteroides fragilis, Clostridium perfringens ( A na-akpọ ya n'ihi njedebe dị nkọ nke nje bacteria), Bacillus tetani, Streptococcus pepticus, Streptococcus pepticus, na JaChemicalbook flagellate. na-ebute ọrịa ọnụ, na 1978 wee mata ya site na World Health Organisation dị ka ọgwụ siri ike megide ọrịa anaerobic ma ejiri ya mee ihe maka mgbochi na ọgwụgwọ nke ọrịa anaerobic ọnụ.A na-ejikwa ya ugboro ugboro n'ụlọ ọgwụ maka mgbochi na ọgwụgwọ nke iku ume, eriri afọ, abdominal na pelvic nje nke nje bacteria anaerobic, akpụkpọ anụ na anụ ahụ dị nro, ọrịa ọkpụkpụ na nkwonkwo, cardiitis, sepsis na ụbụrụ.

2. Usoro nke ime ihe bụ site na nkwụsị nke mmeghachi omume redox nke amoeba protozoa, nke mere na agbụ nitrogen nke protozoa na-agbaji na mmetụta.In vitro ule na-egosi na na ịta nke 1 ~ 2mg / L, morphological mgbanwe nke ameba nke Chemicalbook anụ ahụ nwere ike ime na 6 ~ 20 awa, na ha niile nwere ike igbu n'ime 24 awa.

3.White ma ọ bụ odo odo ma ọ bụ kristal ntụ ntụ;ubé odorous, ilu na ubé nnu.Na-agbaze ntakịrị na ethanol, soluble ntakịrị na mmiri ma ọ bụ chloroform, soluble dị ntakịrị na ether.Methyl Chemicalbook nitrazole bụ ngwakọta heterocyclic nwere nitrogen nwere alkalinity na obere mmiri solubility.Dị ka ụkpụrụ nke premedication si dị, metronidazole na-mere n'ime potassium phosphate nnu, na mmiri solubility na-abawanye, nke a ga-eji dị ka injection ngwọta.

Ngwa

1.Ọ na-eji maka ọgwụgwọ nke trichomoniasis kemgbe 1959 na nsia esịtidem na mpụga amebiasis kemgbe 1970, na elu arụmọrụ, ala toxicity na mbara ngwa.Ọ nwere mmetụta mutagenic na teratogenic na nnwale anụmanụ.
2.Strong antibacterial mmetụta megide ọtụtụ anaerobic bacteria
3.N'ihi na ọgwụgwọ nke amoebiasis, trichomoniasis na anaerobic ọrịa

 


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